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(R)-PR-924

https://www.tbcta.org/web/image/product.template/221824/image_1920?unique=4a1c841
(R)-PR-924 is the isomer of PR-924 (HY-123587), and can be used as an experimental control. PR-924 is a selective tripeptide epoxyketone immunoproteasome subunit LMP-7 inhibitor with an IC50 of 22 nM. PR-924 covalently modifies proteasomal N-terminal threonine active sites. PR-924 inhibits growth and triggers apoptosis in multiple myeloma (MM) cells. PR-924 has antitumor activities.

4.778,80 € 4778.8 EUR 4.778,80 €

4.778,80 €

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